Asymmetric N-Heterocyclic Carbene Catalyzed Annulation of 2-Alkenylbenzothiazoles with α-Chloro Aldehydes

نویسندگان

  • Xiaoxiao Song
  • Qijian Ni
  • Chen Zhu
  • Gerhard Raabe
  • Dieter Enders
چکیده

Diastereo- and enantioselective N-heterocyclic carbene catalyzed 1-azadiene Diels-Alder reactions of (E)-2-styrylbenzothiazoles with α-chloro aldehydes are reported. This annulation strategy provides an efficient access to medicinally important dihydrobenzothiazolopyridin-1-ones in good to excellent yields (44-97%) with very good to excellent stereoselectivities (up to 9:1 dr, 98% ee) and tolerates quite a range of substituents.

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عنوان ژورنال:

دوره 47  شماره 

صفحات  -

تاریخ انتشار 2014